PK parameters= Cmax; Tmax; F: bioavailability; t1/2: half-life; VD: volume of distribution; Cl: clearance; PPB: plasma protein binding;(EQN means that the equation t1/2 = VD / Cl * 0.693 was used
Primary Target and PDB code of Protein-Drug complex
ANTIDIABETIC DIPEPTIDYL-PEPTIDASE IV INHIBITOR HYPOGLYCEMIC AGENTS TYPE 2 DIABETES MELLITUS METABOLISM METABOLITE OF SAXAGLIPTIN IS ONE-HALF AS POTENT AS SAXAGLIPTIN AS DPP4 INHIBITOR
PK parameters= Cmax; Tmax; F: bioavailability; t1/2: half-life; VD: volume of distribution; Cl: clearance; PPB: plasma protein binding;(EQN means that the equation t1/2 = VD / Cl * 0.693 was used
Primary Target and PDB code of Protein-Drug complex
ANTIDIABETIC DIPEPTIDYL-PEPTIDASE IV INHIBITOR HYPOGLYCEMIC AGENTS TYPE 2 DIABETES MELLITUS METABOLISM METABOLITE OF SAXAGLIPTIN IS ONE-HALF AS POTENT AS SAXAGLIPTIN AS DPP4 INHIBITOR