M MACITENTAN (is an active metabolite) | MACITENTAN | ATC C02KX04
CARDIOVASCULAR ANTIHYPERTENSIVE PULMONARY ARTERIAL HYPERTENSION (PAH) ENDOTHELIN RECEPTOR ANTAGONIST ET-1 PREVENTS THE BINDING OF ET-1 TO ITS RECEPTORS ETA AND ETB METABOLITE 20 PERCENT AS POTENT AS THE PARENT DRUG IN VITRO | - | VD 40 LITER PPB 99 PERCENT Cl 0.6 LITER / HOUR (EQN) HT 48 HOUR | ENDOTHELIN RECEPTOR ET-1 | ENDOTHELIN RECEPTOR, ET-A/ET-B ANTAGONIST CHEMBL2096678 ENDOTHELIN RECEPTOR, ET-A/ET-B P24530 ENDOTHELIN B RECEPTOR HOMO SAPIENS MEMBRANE RECEPTOR 7TM1 PEPTIDE SHORT PEPTIDE ENDOTHELIN RECEPTOR | EMA ANSM (in French) Inxight Drugs Dailymed Drugs.com SIDER side effects Chemical Probes Portal ChEMBL BindingDB DrugBank |