M DOLASETRON (is an active metabolite) | DOLASETRON | ATC A04AA04
METABOLISM SEROTONIN 5HT3 ANTAGONIST ANTIEMETIC
| - | Cmax 1.7 MICROMOLAR (200 MILLIGRAM) F 75 PERCENT VD 377 LITER (65 KILOGRAM) PPB 77 PERCENT Cl 52 LITER / HOUR (65 KILOGRAM) HT 8.1 HOUR | 5-HYDROXYTRYPTAMINE 3 RECEPTOR | SEROTONIN 3A (5-HT3A) RECEPTOR ANTAGONIST CHEMBL1899 SEROTONIN 3A (5-HT3A) RECEPTOR P46098 5-HYDROXYTRYPTAMINE RECEPTOR 3A HOMO SAPIENS ION CHANNEL LGIC 5HT3 | EMA ANSM (in French) Inxight Drugs Dailymed Drugs.com SIDER side effects Chemical Probes Portal ChEMBL BindingDB DrugBank |