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1 INNClassRoute (list)PK parameters= Cmax; Tmax; F: bioavailability; t1/2: half-life; VD: volume of distribution; Cl: clearance; PPB: plasma protein binding;(EQN means that the equation t1/2 = VD / Cl * 0.693 was usedPrimary Target and PDB code of Protein-Drug complexTargets from DrugCentral Links
EPINASTINE

EPINASTINE


ATC R06AX24
ATC S01GX10

RESPIRATORY SYSTEM
ANTIHISTAMINE
ANTIALLERGIC
HISTAMINE H1 RECEPTOR ANTAGONISTS

OPHTHALMIC

Cmax 0.16 NANOMOLAR

PPB 64 PERCENT

Cl 56 LITER / HOUR

HT 12 HOUR

HISTAMINE H1 RECEPTOR
5-HYDROXYTRYPTAMINE 2A RECEPTOR
ALPHA-1A ADRENERGIC RECEPTOR
ALPHA-2 ADRENERGIC RECEPTOR

Histamine H1 receptor UNIPROT P35367 HRH1

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