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1 INNClassRoute (list)PK parameters= Cmax; Tmax; F: bioavailability; t1/2: half-life; VD: volume of distribution; Cl: clearance; PPB: plasma protein binding;(EQN means that value was calculated using VD=(Cl*t1/2)/0.693)Primary Target and PDB code of Protein-Drug complexTargets from DrugCentral Links
CARISOPRODOL (has an active metabolite)

CARISOPRODOL


ATC M03BA02
ATC M03BA52
ATC M03BA72

MUSCULO-SKELETAL
MUSCLE RELAXANTS
RELIEVING DISCOMFORT ASSOCIATED WITH CUTE PAINFUL MUSCULOSKELETAL CONDITIONS
ALLOSTERIC EFFECTS ON GABA(A) RECEPTOR (PMID25896767)

ORAL

Cmax 6.92 MICROMOLAR

Tmax 1.7 HOUR

HT 2 HOUR

SOLUBILITY SLIGHTLY SOLUBLE IN WATER

GAMMA-AMINOBUTYRIC-ACID RECEPTOR SUBUNIT ALPHA-1 (GABAA)

Unknown - more at DrugCentralANSM (in French)

Dailymed
Drugs.com

SIDER side effects

Chemical Probes Portal

ChEMBL
BindingDB
DrugBank



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