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1 INNClassRoute (list)PK parameters= Cmax; Tmax; F: bioavailability; t1/2: half-life; VD: volume of distribution; Cl: clearance; PPB: plasma protein binding;(EQN means that value was calculated using VD=(Cl*t1/2)/0.693)Primary Target and PDB code of Protein-Drug complexTargets from DrugCentral Links
RELUGOLIX

RELUGOLIX


ATC H01CC54

HORMONES
TREATMENT OF PROSTATE CANCER
A GONADOTROPIN-RELEASING HORMONE (GNRH) RECEPTOR ANTAGONIST

ORAL

Cmax 344.7 NANOMOLAR

Tmax 2.25 HOUR

F 12 PERCENT

PPB 69.5 PERCENT

Cl 29.4 LITER / HOUR

HT 60.8 HOUR

SOLUBILITY 0.04 MILLIGRAM PER MILLILITER IN WATER

GONADOTROPIN-RELEASING HORMONE (GNRH) RECEPTOR

Unknown - more at DrugCentralANSM (in French)

Dailymed
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SIDER side effects

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ChEMBL
BindingDB
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