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| 1 | INN | Class | Route (list) | PK parameters= Cmax; Tmax; F: bioavailability; t1/2: half-life; VD: volume of distribution; Cl: clearance; PPB: plasma protein binding;(EQN means that value was calculated using VD=(Cl*t1/2)/0.693) | Primary Target and PDB code of Protein-Drug complex | Targets from DrugCentral | Links | |||
| RELUGOLIX
| RELUGOLIX | HORMONES | ORAL | Cmax 344.7 NANOMOLAR Tmax 2.25 HOUR F 12 PERCENT PPB 69.5 PERCENT Cl 29.4 LITER / HOUR HT 60.8 HOUR SOLUBILITY 0.04 MILLIGRAM PER MILLILITER IN WATER | GONADOTROPIN-RELEASING HORMONE (GNRH) RECEPTOR | Gonadotropin-releasing hormone receptor UNIPROT P30968 GNRHR more at DrugCentral | EMA | |||
