SAMIDORPHAN 
| SAMIDORPHAN | NERVOUS SYSTEM TREATMENT OF SCHIZOPHRENIA OR BIPOLAR I DISORDER OPIOID RECEPTOR ANTAGONIST OR PARTIAL AGONIST N-DEALKYLATED AND N-OXIDE ARE ACTIVE METABOLITES BUT THEY DO NOT HAVE CAS NUMBER THUS NOT YET INCLUDED HERE | ORAL | Cmax 121.7 NANOMOLAR Tmax 1.5 HOUR F 69 PERCENT PPB 28 PERCENT Cl 40 LITER / HOUR HT 9 HOUR | MU-OPIOID RECEPTOR (KI=0.052 NANOMOLAR) KAPPA-OPIOID RECEPTOR (KI=0.23 NANOMOLAR) DELTA-OPIOID RECEPTOR (KI=2.7 NANOMOLAR) | Unknown - more at DrugCentral | ANSM (in French) Dailymed Drugs.com SIDER side effects Chemical Probes Portal ChEMBL BindingDB DrugBank |