M APALUTAMIDE (is an active metabolite) 
| APALUTAMIDE | ATC L02BB05
ANTINEOPLASTIC ANDROGEN RECEPTOR INHIBITOR INDICATED FOR THE TREATMENT OF PATIENTS WITH NON-METASTATIC CASTRATION-RESISTANT PROSTATE CANCER N-DESMETHYL APALUTAMIDE, IS A LESS POTENT INHIBITOR OF AR, AND EXHIBITED ONE-THIRD THE ACTIVITY | - | Cmax 12.7 MICROMOLAR PPB 95 PERCENT | ANDROGEN RECEPTOR | NUCLEAR RECEPTOR ANDR_HUMAN INHIBITOR P10275 | ANSM (in French) Dailymed Drugs.com SIDER side effects Chemical Probes Portal ChEMBL BindingDB DrugBank |