PK parameters= Cmax; Tmax; F: bioavailability; t1/2: half-life; VD: volume of distribution; Cl: clearance; PPB: plasma protein binding;(EQN means that the equation t1/2 = VD / Cl * 0.693 was used
Primary Target and PDB code of Protein-Drug complex
PK parameters= Cmax; Tmax; F: bioavailability; t1/2: half-life; VD: volume of distribution; Cl: clearance; PPB: plasma protein binding;(EQN means that the equation t1/2 = VD / Cl * 0.693 was used
Primary Target and PDB code of Protein-Drug complex
CARDIOVASCULAR HYPOLIPIDEMIC ANTICHOLESTEREMIC AGENTS ANTILIPIDEMIC AGENTS REDUCE THE VERY LOW-DENSITY LIPOPROTEIN FRACTION
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Cmax 932.8 MICROMOLAR
PPB 96 PERCENT
HT 20 HOUR
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTOR
PDB7BPY (X-RAY STRUCTURE OF HUMAN PPARALPHA LIGAND BINDING DOMAIN-CLOFIBRIC ACID-SRC1 COACTIVATOR PEPTIDE CO-CRYSTALS OBTAINED BY DELIPIDATION AND CO-CRYSTALLIZATION)