| M TETRABENAZINE                                                                                                                                                                                                                                                   (is an active metabolite)  
  |  TETRABENAZINE |  ATC N07XX06
  NERVOUS SYSTEM   CNS   TREATMENT OF CHOREA ASSOCIATED WITH HUNTINGTON DISEASE   INHIBITOR   IS BELIEVED TO BE RELATED TO ITS EFFECT AS A REVERSIBLE DEPLETOR OF MONOAMINES (SUCH AS DOPAMINE, SEROTONIN, NOREPINEPHRINE, AND HISTAMINE) FROM NERVE TERMINALS   VESICULAR MONOAMINE TRANSPORTER TYPE 2 (VMAT2) (KI=100 NANOMOLAR)  | - | Tmax 1 HOUR PPB 61 PERCENT HT 5 HOUR  |  VESICULAR MONOAMINE TRANSPORTER TYPE 2 (VMAT2) |   Synaptic vesicular amine transporter UNIPROT Q05940 SLC18A2  more at DrugCentral  | EMA ANSM (in French) Inxight Drugs Dailymed Drugs.com VigiAccess SIDER side effects Chemical Probes Portal ChEMBL BindingDB DrugBank  |