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1 INNClassRoute (list)PK parameters= Cmax; Tmax; F: bioavailability; t1/2: half-life; VD: volume of distribution; Cl: clearance; PPB: plasma protein binding;(EQN means that value was calculated using VD=(Cl*t1/2)/0.693)Primary Target and PDB code of Protein-Drug complexTargets from DrugCentral Links
PARICALCITOL

PARICALCITOL


ATC A11CC07
ATC H05BX02

METABOLISM
PARATHYROID HORMONE REGULATOR
VITAMIN D3 RECEPTOR (VDR) AGONIST
CALCITRIOL ANALOG
TREATMENT OF SECONDARY HYPERPARATHYROIDISM

INTRAVENOUS ORAL INJECTION

Cmax 4.03 NANOMOLAR

F 79 PERCENT

VD 34 LITER

PPB 99.8 PERCENT

Cl 1.49 LITER / HOUR

HT 5 HOUR

VITAMIN D3 RECEPTOR

VITAMIN D RECEPTOR AGONIST CHEMBL1977 VITAMIN D RECEPTOR P11473 VITAMIN D3 RECEPTOR HOMO SAPIENS TRANSCRIPTION FACTOR NUCLEAR RECEPTOR NR1 NR1I NR1I1EMA

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