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1 INNClassRoute (list)PK parameters= Cmax; Tmax; F: bioavailability; t1/2: half-life; VD: volume of distribution; Cl: clearance; PPB: plasma protein binding;(EQN means that value was calculated using VD=(Cl*t1/2)/0.693)Primary Target and PDB code of Protein-Drug complexTargets from DrugCentral Links
CERIVASTATIN DISCONTINUED

CERIVASTATIN


ATC C10AA06

CARDIOVASCULAR
HYPOCHOLESTEROLEMIC
3-HYDROXY-3-METHYLGLUTARYL-COENZYME A REDUCTASE (HMG-COA) INHIBITOR
ANTI-LIPIDEMIC AGENTS

ORAL

Cmax 27.6 MICROMOLAR

Tmax 2 HOUR

F 60 PERCENT

VD 19.5 LITER (65 KILOGRAM)

PPB 99 PERCENT

Cl 12.5 LITER / HOUR

HT 3 HOUR

SOLUBILITY SOLUBLE IN WATER

3-HYDROXY-3-METHYLGLUTARYL-COENZYME A REDUCTASE

HMG-COA REDUCTASE INHIBITOR CHEMBL402 HMG-COA REDUCTASE P04035 3-HYDROXY-3-METHYLGLUTARYL-COENZYME A REDUCTASE HOMO SAPIENS ENZYME REDUCTASEEMA

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