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1 INNClassRoute (list)PK parameters= Cmax; Tmax; F: bioavailability; t1/2: half-life; VD: volume of distribution; Cl: clearance; PPB: plasma protein binding;(EQN means that value was calculated using VD=(Cl*t1/2)/0.693)Primary Target and PDB code of Protein-Drug complexTargets from DrugCentral Links
CISAPRIDE DISCONTINUED

CISAPRIDE


ATC A03FA02

METABOLISM
GASTROINTESTINAL AGENTS
TREATMENT OF NOCTURNAL HEARTBURN DUE TO GASTROESOPHAGEAL REFLUX DISEASE
SEROTONIN RECEPTOR 5-HT4 AGONIST

ORAL

Tmax 1.25 HOUR

F 37.5 PERCENT

VD 180 LITER

PPB 98 PERCENT

Cl 6 LITER / HOUR

HT 4 HOUR

SOLUBILITY PRACTICALLY INSOLUBLE IN WATER

5-HYDROXYTRYPTAMINE 4 RECEPTOR

SEROTONIN 4 (5-HT4) RECEPTOR AGONIST CHEMBL1875 SEROTONIN 4 (5-HT4) RECEPTOR Q13639 5-HYDROXYTRYPTAMINE RECEPTOR 4 HOMO SAPIENS MEMBRANE RECEPTOR 7TM1 SMALLMOL MONOAMINE RECEPTOR SEROTONIN RECEPTOREMA

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