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1 INNClassRoute (list)PK parameters= Cmax; Tmax; F: bioavailability; t1/2: half-life; VD: volume of distribution; Cl: clearance; PPB: plasma protein binding;(EQN means that value was calculated using VD=(Cl*t1/2)/0.693)Primary Target and PDB code of Protein-Drug complexTargets from DrugCentral Links
CLOFAZIMINE DISCONTINUED

CLOFAZIMINE


ATC J04BA01

ANTIINFECTIVES
ANTIMYCOBACTERIALS
LEPROSTATIC AGENTS
ANTI-INFLAMMATORY
TREATMENT OF LEPROMATOUS LEPROSY

ORAL

Cmax 2.1 MICROMOLAR (300 MILLIGRAM)

Tmax 10 HOUR

F 53 PERCENT

HT 1680 HOUR

SOLUBILITY INSOLUBLE IN WATER

DNA

DNA INHIBITOR CHEMBL2366041 DNA MYCOBACTERIUM LEPRAEEMA

ANSM (in French)

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