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1 INNClassRoute (list)PK parameters= Cmax; Tmax; F: bioavailability; t1/2: half-life; VD: volume of distribution; Cl: clearance; PPB: plasma protein binding;(EQN means that value was calculated using VD=(Cl*t1/2)/0.693)Primary Target and PDB code of Protein-Drug complexTargets from DrugCentral Links
DIAZOXIDE

DIAZOXIDE


ATC C02DA01
ATC V03AH01

CARDIOVASCULAR
ANTIHYPERTENSIVE
NONDIURETIC BENZOTHIADIAZINE
VASODILATOR AGENTS
MANAGEMENT OF SYMPTOMATIC HYPOGLYCEMIA
INCREASE IN BLOOD GLUCOSE LEVEL SELECTIVE MITOCHONDRIAL KATP-CHANNEL AGONIST

INJECTION ORAL

Tmax 1 HOUR

VD 13.6 LITER (65 KILOGRAM)

PPB 94 PERCENT

Cl 0.23 LITER / HOUR (65 KILOGRAM)

HT 48 HOUR

SOLUBILITY SPARINGLY SOLUBLE IN WATER

MITOCHONDRIAL KATP-CHANNEL (PMID9400389)

SODIUM/POTASSIUM-TRANSPORTING ATPASE SUBUNIT ALPHA-1 P05023 SODIUM/POTASSIUM-TRANSPORTING ATPASE SUBUNIT ALPHA-1 HOMO SAPIENS ENZYME HYDROLASEEMA

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