TELOTRISTAT ETHYL (has an active metabolite) | TELOTRISTAT ETHYL | ATC A16AX15
METABOLISM TREATMENT OF CARCINOID SYNDROME DIARRHEA TRYPTOPHAN HYDROXYLASE INHIBITOR WHICH MEDIATES THE RATE LIMITING STEP IN SEROTONIN BIOSYNTHESIS | ORAL | Cmax 7.6 NANOMOLAR Tmax 1.25 HOUR PPB 99 PERCENT Cl 2.7 LITER / HOUR HT 0.6 HOUR SOLUBILITY NEGLIGIBLE AT A PH OF 5 TO 9 | TRYPTOPHAN HYDROXYLASE | ENZYME TPH1_HUMAN INHIBITOR P17752 | EMA ANSM (in French) Inxight Drugs Dailymed Drugs.com SIDER side effects Chemical Probes Portal ChEMBL BindingDB DrugBank |