LUMACAFTOR | LUMACAFTOR | ATC R07AX30
RESPIRATORY SYSTEM CYSTIC FIBROSIS POTENTIATOR IMPROVES THE CONFORMATIONAL STABILITY OF F508DEL-CFTR RESULTING IN INCREASED PROCESSING AND TRAFFICKING OF MATURE PROTEIN TO THE CELL SURFACE | ORAL | Cmax 55.3 MICROMOLAR Tmax 4 HOUR VD 86 LITER PPB 99 PERCENT Cl 2.38 LITER / HOUR HT 25.2 HOUR SOLUBILITY PRACTICALLY INSOLUBLE IN WATER | CFTR CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR | CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR STABILISER CHEMBL4051 CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR P13569 CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR HOMO SAPIENS ION CHANNEL OTHER CHLORIDE CFTR | EMA ANSM (in French) Inxight Drugs Dailymed Drugs.com SIDER side effects Chemical Probes Portal ChEMBL BindingDB DrugBank |