LURASIDONE | LURASIDONE | ATC N05AE05
NERVOUS SYSTEM ANTIPSYCHOTIC SCHIZOPHRENIA OF BENZISOTHIAZOL DERIVATIVES ANTAGONIST | ORAL | VD 6173 LITER (40 MILLIGRAM) PPB 99 PERCENT Cl 234 LITER / HOUR (40 MILLIGRAM) HT 18 HOUR (40 MILLIGRAM) SOLUBILITY VERY SLIGHTLY SOLUBLE IN WATER | DOPAMINE D2 ANTAGONIST (KI=0.994 NANOMOLAR) 5-HT2A ANTAGONIST (KI=0.47 NANOMOLAR) 5-HT7 ANTAGONIST (KI=0.495 NANOMOLAR) ALPHA2C-ADRENERGIC RECEPTOR ANTAGONIST (KI=10.8 NANOMOLAR) 5-HT1A RECEPTOR PARTIAL AGONIST (KI=6.38 NANOMOLAR) ALPHA2A ADRENERGIC RECEPTORS ANTAGONIST (KI=40.7 NM) | DOPAMINE D2 RECEPTOR ANTAGONIST CHEMBL217 DOPAMINE D2 RECEPTOR P14416 D(2) DOPAMINE RECEPTOR HOMO SAPIENS MEMBRANE RECEPTOR 7TM1 SMALLMOL MONOAMINE RECEPTOR DOPAMINE RECEPTOR | EMA ANSM (in French) Inxight Drugs Dailymed Drugs.com SIDER side effects Chemical Probes Portal ChEMBL BindingDB DrugBank |