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1 INNClassRoute (list)PK parameters= Cmax; Tmax; F: bioavailability; t1/2: half-life; VD: volume of distribution; Cl: clearance; PPB: plasma protein binding;(EQN means that value was calculated using VD=(Cl*t1/2)/0.693)Primary Target and PDB code of Protein-Drug complexTargets from DrugCentral Links
ERGOLOID

ERGOLOID


ATC C04AE01
ATC C04AE51

CARDIOVASCULAR
COGNITION ENHANCER
ADRENERGIC ALPHA ANTAGONISTS
NOOTROPIC AGENTS
SYMPATHOLYTICS (PMID9787282)

SUBLINGUAL ORAL

Tmax 2.25 HOUR

F 50 PERCENT

HT 3.85 HOUR

ALPHA ADRENERGIC RECEPTOR

SEROTONIN 1A (5-HT1A) RECEPTOR AGONIST CHEMBL214 SEROTONIN 1A (5-HT1A) RECEPTOR P08908 5-HYDROXYTRYPTAMINE RECEPTOR 1A HOMO SAPIENS MEMBRANE RECEPTOR 7TM1 SMALLMOL MONOAMINE RECEPTOR SEROTONIN RECEPTOREMA

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