BACLOFEN | BACLOFEN | ATC M03BX01
MUSCULO-SKELETAL SYSTEM MUSCLE RELAXANT GABA AGONISTS | ORAL INTRATHECAL | VD 59 LITER PPB 30 PERCENT Cl 10 LITER / HOUR HT 5 HOUR SOLUBILITY SLIGHTLY SOLUBLE IN WATER | GAMMA-AMINOBUTYRIC ACID TYPE B RECEPTOR PDB 4MS4 (CRYSTAL STRUCTURE OF THE EXTRACELLULAR DOMAIN OF HUMAN GABA(B) RECEPTOR BOUND TO THE AGONIST BACLOFEN) LIGAND CODE = 2C0 (link to the list of PDB complexes) Download experimental 3D coordinates of 2C0 with added hydrogens | GABA-B RECEPTOR AGONIST CHEMBL2111463 GABA-B RECEPTOR O75899 GAMMA-AMINOBUTYRIC ACID TYPE B RECEPTOR SUBUNIT 2 HOMO SAPIENS MEMBRANE RECEPTOR 7TM3 SMALLMOL NEUROTRANSMITTER GABA-B RECEPTOR | EMA ANSM (in French) Inxight Drugs Dailymed Drugs.com SIDER side effects Chemical Probes Portal ChEMBL BindingDB DrugBank |