BORTEZOMIB | BORTEZOMIB | ATC L01XX32
ANTINEOPLASTIC AGENTS PROTEASE INHIBITORS COVALENT BUT REVERSIBLE INHIBITOR | INTRAVENOUS SUBCUTANEOUS INJECTION | Cmax 321.7 NANOMOLAR VD 1917 LITER PPB 83 PERCENT Cl 32 LITER / HOUR HT 92 HOUR | 26S PROTEASOME PDB 4QW1 (YCP BETA5-A50V MUTANT IN COMPLEX WITH BORTEZOMIB) LIGAND CODE = BO2 (link to the list of PDB complexes) Download experimental 3D coordinates of BO2 with added hydrogens | 26S PROTEOSOME INHIBITOR CHEMBL2364701 26S PROTEOSOME P28074 PROTEASOME SUBUNIT BETA HOMO SAPIENS ENZYME PROTEASE THREONINE PBT T1A | EMA ANSM (in French) Inxight Drugs Dailymed Drugs.com SIDER side effects Chemical Probes Portal ChEMBL BindingDB DrugBank |