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1 INNClassRoute (list)PK parameters= Cmax; Tmax; F: bioavailability; t1/2: half-life; VD: volume of distribution; Cl: clearance; PPB: plasma protein binding;(EQN means that value was calculated using VD=(Cl*t1/2)/0.693)Primary Target and PDB code of Protein-Drug complexTargets from DrugCentral Links
TROSPIUM

TROSPIUM


ATC G04BD09
ATC A03DA06

METABOLISM
ANTISPASMODIC
ANTICHOLINERGIC
ANALGESICS
PARASYMPATHOLYTICS

ORAL

Cmax 8.9 NANOMOLAR

Tmax 5.5 HOUR

F 9.6 PERCENT

VD 395 LITER

PPB 67 PERCENT

Cl 13.6 LITER / HOUR (EQN)

HT 20 HOUR

SOLUBILITY 1 GRAM / 2 MILLILITER

MUSCARINIC ACETYLCHOLINE RECEPTOR M1

MUSCARINIC ACETYLCHOLINE RECEPTOR M2 ANTAGONIST CHEMBL211 MUSCARINIC ACETYLCHOLINE RECEPTOR M2 P08172 MUSCARINIC ACETYLCHOLINE RECEPTOR M2 HOMO SAPIENS MEMBRANE RECEPTOR 7TM1 SMALLMOL MONOAMINE RECEPTOR ACETYLCHOLINE RECEPTOREMA

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