| | ||||||||||
| 1 | INN | Class | Route (list) | PK parameters= Cmax; Tmax; F: bioavailability; t1/2: half-life; VD: volume of distribution; Cl: clearance; PPB: plasma protein binding;(EQN means that value was calculated using VD=(Cl*t1/2)/0.693) | Primary Target and PDB code of Protein-Drug complex | Targets from DrugCentral | Links | |||
| CETRORELIX
| CETRORELIX | HORMONES | SUBCUTANEOUS | Cmax 19.9 NANOMOLAR Tmax 1.5 HOUR F 85 PERCENT VD 75.4 LITER (65 KILOGRAM) PPB 86 PERCENT Cl 5 LITER / HOUR (65 KILOGRAM) HT 62.8 HOUR | GONADOTROPIN-RELEASING HORMONE RECEPTOR | GONADOTROPIN-RELEASING HORMONE RECEPTOR ANTAGONIST CHEMBL1855 GONADOTROPIN-RELEASING HORMONE RECEPTOR P30968 GONADOTROPIN-RELEASING HORMONE RECEPTOR HOMO SAPIENS MEMBRANE RECEPTOR 7TM1 PEPTIDE SHORT PEPTIDE GNRH RECEPTOR | EMA | |||
