ZALEPLON | ZALEPLON | ATC N05CF03
NERVOUS SYSTEM HYPNOTIC ANXIOLYTIC ANTICONVULSANTS MUSCLE RELAXANT SEDATIVE A NONBENZODIAZEPINE HYPNOTIC FROM THE PYRAZOLOPYRIMIDINE | ORAL | Cmax 980 NANOMOLAR (PMID18621671) Tmax 1 HOUR F 30 PERCENT VD 91 LITER (65 KILOGRAM) PPB 60 PERCENT Cl 195 LITER / HOUR (65 KILOGRAM) HT 1 HOUR SOLUBILITY PRACTICALLY INSOLUBLE IN WATER | GAMMA-AMINOBUTYRIC-ACID RECEPTOR (GABA) BRAIN OMEGA-1 RECEPTOR | GABA A RECEPTOR ALPHA-1/BETA-1/GAMMA-2 POSITIVE ALLOSTERIC MODULATOR CHEMBL2111392 GABA A RECEPTOR ALPHA-1/BETA-1/GAMMA-2 P18505 GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT BETA-1 HOMO SAPIENS ION CHANNEL LGIC GABAA | EMA ANSM (in French) Inxight Drugs Dailymed Drugs.com SIDER side effects Chemical Probes Portal ChEMBL BindingDB DrugBank |