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1 INNClassRoute (list)PK parameters= Cmax; Tmax; F: bioavailability; t1/2: half-life; VD: volume of distribution; Cl: clearance; PPB: plasma protein binding;(EQN means that value was calculated using VD=(Cl*t1/2)/0.693)Primary Target and PDB code of Protein-Drug complexTargets from DrugCentral Links
CISATRACURIUM

CISATRACURIUM
ATRACURIUM


ATC M03AC11

METABOLISM
NEUROMUSCULAR BLOCKER
NONDEPOLARIZING SKELETAL MUSCLE RELAXANT
CHOLINERGIC RECEPTORS ANTAGONISTS

INJECTION

VD 9.4 LITER (65 KILOGRAM)

PPB 38 PERCENT

Cl 17.8 LITER / HOUR (65 KILOGRAM)

HT 0.36 HOUR

SOLUBILITY LOGP=-2.12

ACETYLCHOLINE RECEPTOR SUBUNIT ALPHA-2

MUSCLE-TYPE NICOTINIC ACETYLCHOLINE RECEPTOR ANTAGONIST CHEMBL2362997 MUSCLE-TYPE NICOTINIC ACETYLCHOLINE RECEPTOR P02708 ACETYLCHOLINE RECEPTOR SUBUNIT ALPHA HOMO SAPIENS ION CHANNEL LGIC ACH CHRN ALPHAEMA

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