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1 INNClassRoute (list)PK parameters= Cmax; Tmax; F: bioavailability; t1/2: half-life; VD: volume of distribution; Cl: clearance; PPB: plasma protein binding;(EQN means that value was calculated using VD=(Cl*t1/2)/0.693)Primary Target and PDB code of Protein-Drug complexTargets from DrugCentral Links
MORICIZINE DISCONTINUED

MORICIZINE


ATC C01BG01

CARDIOVASCULAR
ANTIARRHYTHMIC

ORAL

Cmax 2.3 MICROMOLAR (2.2 MILLIGRAM / KILOGRAM) (PMID8568009)

Tmax 0.8 HOUR

F 36 PERCENT

VD 300 LITER (PMID8568009)

PPB 93.5 PERCENT (PMID8568009)

Cl 150 LITER / HOUR (PMID10434234)

HT 1.9 HOUR

SODIUM CHANNEL

SODIUM CHANNEL ALPHA SUBUNIT BLOCKER CHEMBL2331043 SODIUM CHANNEL ALPHA SUBUNIT P35498 SODIUM CHANNEL PROTEIN TYPE 1 SUBUNIT ALPHA HOMO SAPIENS ION CHANNEL VGC VG NAEMA

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