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1 INNClassRoute (list)PK parameters= Cmax; Tmax; F: bioavailability; t1/2: half-life; VD: volume of distribution; Cl: clearance; PPB: plasma protein binding;(EQN means that value was calculated using VD=(Cl*t1/2)/0.693)Primary Target and PDB code of Protein-Drug complexTargets from DrugCentral Links
METYROSINE

METYROSINE


ATC C02KB01

ANTIHYPERTENSIVE
TREATMENT OF PHEOCHROMOCYTOMA (TUMOR OF THE ADRENAL GLAND)
DECREASES ENDOGENOUS LEVELS OF CATECHOLAMINES

ORAL

F 69 PERCENT

HT 3.3 HOUR

SOLUBILITY VERY SLIGHTLY SOLUBLE IN WATER

TYROSINE HYDROXYLASE

TYROSINE 3-HYDROXYLASE INHIBITOR CHEMBL1969 TYROSINE 3-HYDROXYLASE P07101 TYROSINE 3-MONOOXYGENASE HOMO SAPIENS ENZYME REDUCTASEEMA

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