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1 INNClassRoute (list)PK parameters= Cmax; Tmax; F: bioavailability; t1/2: half-life; VD: volume of distribution; Cl: clearance; PPB: plasma protein binding;(EQN means that value was calculated using VD=(Cl*t1/2)/0.693)Primary Target and PDB code of Protein-Drug complexTargets from DrugCentral Links
CHLORPROTHIXENE DISCONTINUED

CHLORPROTHIXENE


ATC N05AF03

NERVOUS SYSTEM
ANTIPSYCHOTIC
DOPAMINE D2 ANTAGONISTS

ORAL INJECTION

Cmax 1.36 MICROMOLAR

Tmax 4 HOUR

F 17 PERCENT (PMID10525070)

VD 1035 LITER

Cl 52 LITER / HOUR

HT 25.8 HOUR

D(2) DOPAMINE RECEPTOR

DOPAMINE D2 RECEPTOR ANTAGONIST CHEMBL217 DOPAMINE D2 RECEPTOR P14416 D(2) DOPAMINE RECEPTOR HOMO SAPIENS MEMBRANE RECEPTOR 7TM1 SMALLMOL MONOAMINE RECEPTOR DOPAMINE RECEPTOREMA

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