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1 INNClassRoute (list)PK parameters= Cmax; Tmax; F: bioavailability; t1/2: half-life; VD: volume of distribution; Cl: clearance; PPB: plasma protein binding;(EQN means that value was calculated using VD=(Cl*t1/2)/0.693)Primary Target and PDB code of Protein-Drug complexTargets from DrugCentral Links
BIPERIDEN DISCONTINUED

BIPERIDEN


ATC N04AA02

NERVOUS SYSTEM
ANTIPARKINSONIAN
PERIPHERAL ANTICHOLINERGIC
ANTISPASMODIC
ANTIDYSKINETICS
MUSCARINIC ANTAGONISTS
PARASYMPATHOLYTICS

ORAL INJECTION

Cmax 16 NANOMOLAR

Tmax 1.25 HOUR

VD 780 LITER (65 KILOGRAM)

PPB 90 PERCENT

Cl 46.8 LITER / HOUR (65 KILOGRAM)

HT 24 HOUR

SOLUBILITY SLIGHTLY SOLUBLE IN WATER

MUSCARINIC ACETYLCHOLINE RECEPTOR

MUSCARINIC ACETYLCHOLINE RECEPTOR M1 ANTAGONIST CHEMBL216 MUSCARINIC ACETYLCHOLINE RECEPTOR M1 P11229 MUSCARINIC ACETYLCHOLINE RECEPTOR M1 HOMO SAPIENS MEMBRANE RECEPTOR 7TM1 SMALLMOL MONOAMINE RECEPTOR ACETYLCHOLINE RECEPTOREMA

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