AVAPRITINIB | AVAPRITINIB | ATC L01EX18
ANTINEOPLASTIC A TYROSINE KINASE INHIBITOR PDGFRA AND PDGFRA D842 MUTANTS AND KIT TREATMENT OF UNRESECTABLE OR METASTATIC GASTROINTESTINAL STROMAL TUMOR (GIST) | ORAL | Cmax 1.63 MICROMOLAR Tmax 3 HOUR VD 1200 LITER PPB 98.8 PERCENT Cl 19.5 LITER / HOUR HT 44.5 HOUR SOLUBILITY LOWER THAN 0.001 MILLIGRAM PER MILLILITER | PLATELET-DERIVED GROWTH FACTOR RECEPTOR ALPHA (PDGFRA) MAST STEM CELL GROWTH FACTOR RECEPTOR (KIT) | Platelet-derived growth factor receptor alpha inhibitor P16234 (PGFRA_HUMAN) | EMA ANSM (in French) Inxight Drugs Dailymed Drugs.com SIDER side effects Chemical Probes Portal ChEMBL BindingDB DrugBank |