PEXIDARTINIB | PEXIDARTINIB | ATC L01EX15
ANTINEOPLASTIC TYROSINE KINASE INHIBITOR COLONY STIMULATING ACTOR 1 RECEPTOR (CSF1R), KIT PROTO-ONCOGENE RECEPTOR TYROSINE KINASE (KIT), AND FMS-LIKE TYROSINE KINASE 3 (FLT3) TREATMENT OF SYMPTOMATIC TENOSYNOVIAL GIANT CELL TUMOR (TGCT) | ORAL | Cmax 20.6 MICROMOLAR Tmax 2.5 HOUR VD 187 LITER PPB 99 PERCENT Cl 5.1 LITER / HOUR HT 26.6 HOUR SOLUBILITY SLIGHTLY SOLUBLE IN WATER | COLONY STIMULATING ACTOR 1 RECEPTOR (CSF1R) PDB 4R7H (CRYSTAL STRUCTURE OF FMS KINASE DOMAIN WITH A SMALL MOLECULAR INHIBITOR, PLX3397) LIGAND CODE = P31 (link to the list of PDB complexes) Download experimental 3D coordinates of P31 with added hydrogens | Macrophage colony-stimulating factor 1 receptor INHIBITOR P07333 CSF1R_HUMAN | EMA ANSM (in French) Inxight Drugs Dailymed Drugs.com SIDER side effects Chemical Probes Portal ChEMBL BindingDB DrugBank |