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1 INNClassRoute (list)PK parameters= Cmax; Tmax; F: bioavailability; t1/2: half-life; VD: volume of distribution; Cl: clearance; PPB: plasma protein binding;(EQN means that value was calculated using VD=(Cl*t1/2)/0.693)Primary Target and PDB code of Protein-Drug complexTargets from DrugCentral Links
TENAPANOR

TENAPANOR


ATC A06AX08

NERVOUS SYSTEM
SODIUM/HYDROGEN EXCHANGER 3 (NHE3) INHIBITOR
TREATMENT OF IRRITABLE BOWEL SYNDROME WITH CONSTIPATION (IBS-C)

ORAL

PPB 99 PERCENT

SOLUBILITY PRACTICALLY INSOLUBLE IN WATER

SODIUM/HYDROGEN EXCHANGER 3 (NHE3)

transporter Sodium/hydrogen exchanger 3 inhibitor P48764 SL9A3_HUMANEMA

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