ENCORAFENIB | ENCORAFENIB | ATC L01XE46
ANTINEOPLASTIC BRAF V600E KINASE INHIBITOR (KD=0.35 NANOMOLAR) TREATMENT OF MELANOMA WITH A BRAF V600E OR V600K MUTATION ALSO BINDS JNK1, JNK2, JNK3, LIMK1, LIMK2, MEK4, AND STK36 KINASES | ORAL | Tmax 2 HOUR F 86 PERCENT VD 164 LITER PPB 86 PERCENT Cl 14 LITER / HOUR HT 3.5 HOUR SOLUBILITY INSOLUBLE IN WATER AT PH 3 AND HIGHER | BRAF | Serine/threonine-protein kinase B-raf P15056 | EMA ANSM (in French) Inxight Drugs Dailymed Drugs.com SIDER side effects Chemical Probes Portal ChEMBL BindingDB DrugBank |