COPANLISIB | COPANLISIB | ATC L01XX61
ANTINEOPLASTIC PHOSPHATIDYLINOSITOL-3-KINASE (PI3K) INHIBITOR WITH INHIBITORY ACTIVITY PREDOMINANTLY AGAINST PI3K-ALPHA AND PI3K-DELTA ISOFORMS EXPRESSED IN MALIGNANT B CELLS TREATMENT OF FOLLICULAR LYMPHOMA | INTRAVENOUS | Cmax 964 NANOMOLAR VD 871 LITER PPB 84.2 PERCENT Cl 17.9 LITER / HOUR HT 39.1 HOUR | PHOSPHATIDYLINOSITOL-3-KINASE (PI3K) PDB 5G2N (X-RAY STRUCTURE OF PI3KINASE GAMMA IN COMPLEX WITH COPANLISIB) LIGAND CODE = 6E2 (link to the list of PDB complexes) Download experimental 3D coordinates of 6E2 with added hydrogens | KINASE PK3CA_HUMAN INHIBITOR P42336 PK3CD_HUMAN INHIBITOR O00329 | EMA ANSM (in French) Inxight Drugs Dailymed Drugs.com SIDER side effects Chemical Probes Portal ChEMBL BindingDB DrugBank |