M CARBAMAZEPINE (is an active metabolite) | CARBAMAZEPINE | ATC N03AF01
NERVOUS SYSTEM ANTICONVULSANT ANALGESIC ANTIMANIC AGENTS SPECIFIC ANALGESIC FOR TRIGEMINAL NEURALGIA CARBAMAZEPINE INDUCES ITS OWN METABOLISM MECHANISM OF ACTION UNKNOWN (NUMEROUS PHARMACOLOGICAL EFFECTS HAVE BEEN DESCRIBED MODULATION OF ION CHANNELS (SODIUM AND CALCIUM), RECEPTOR-MEDIATED NEUROTRANSMISSION (GABAERGIC, GLUTAMATERGIC, AND MONOAMINERGIC), AND INTRACELLULAR SIGNALING PATHWAYS) | - | Cmax 8.7 MICROMOLAR Tmax 14 HOUR PPB 50 PERCENT HT 34 HOUR | VOLTAGE-GATED SODIUM CHANNELS | NEURONAL ACETYLCHOLINE RECEPTOR ALPHA2/BETA4 P30926 NEURONAL ACETYLCHOLINE RECEPTOR SUBUNIT BETA-4 HOMO SAPIENS ION CHANNEL LGIC ACH CHRN BETA | EMA ANSM (in French) Inxight Drugs Dailymed Drugs.com SIDER side effects Chemical Probes Portal ChEMBL BindingDB DrugBank |