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1 INNClassRoute (list)PK parameters= Cmax; Tmax; F: bioavailability; t1/2: half-life; VD: volume of distribution; Cl: clearance; PPB: plasma protein binding;(EQN means that value was calculated using VD=(Cl*t1/2)/0.693)Primary Target and PDB code of Protein-Drug complexTargets from DrugCentral Links
DAPAGLIFLOZIN

DAPAGLIFLOZIN


ATC A10BX09
ATC A10BD15
ATC A10BK01
ATC A10BD25
ATC A10BD21

METABOLISM
A SODIUM-GLUCOSE COTRANSPORTER 2 (SGLT2) INHIBITOR
TREATMENT OF TYPE 2 DIABETES MELLITU
IMPROVE GLYCEMIC CONTROL

ORAL

Tmax 2 HOUR

F 78 PERCENT

PPB 91 PERCENT

HT 12.9 HOUR

SODIUM-GLUCOSE COTRANSPORTER 2 (SGLT2)

SODIUM/GLUCOSE COTRANSPORTER 2 INHIBITOR CHEMBL3884 SODIUM/GLUCOSE COTRANSPORTER 2 P31639 SODIUM/GLUCOSE COTRANSPORTER 2 HOMO SAPIENS TRANSPORTER ELECTROCHEMICAL SLC SLC05EMA

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