REGORAFENIB | REGORAFENIB | ATC L01XE21
ANTINEOPLASTIC METASTATIC COLORECTAL CANCER KINASES INHIBITOR | ORAL | Cmax 5.1 MICROMOLAR Tmax 4 HOUR F 76 PERCENT PPB 99.5 PERCENT HT 28 HOUR SOLUBILITY PRACTICALLY INSOLUBLE IN WATER | RET VEGFR1 VEGFR2 VEGFR3 KIT PDGFR-ALPHA PDGFR-BETA FGFR1 FGFR2 TIE2 DDR2 TRK2A EPH2A RAF-1 BRAF BRAF(V600E) SAPK2 PTK5 ABL | TYROSINE-PROTEIN KINASE ABL INHIBITOR CHEMBL1862 TYROSINE-PROTEIN KINASE ABL P00519 TYROSINE-PROTEIN KINASE ABL1 HOMO SAPIENS ENZYME KINASE PROTEIN KINASE TK ABL | EMA ANSM (in French) Inxight Drugs Dailymed Drugs.com SIDER side effects Chemical Probes Portal ChEMBL BindingDB DrugBank |