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1 INNClassRoute (list)PK parameters= Cmax; Tmax; F: bioavailability; t1/2: half-life; VD: volume of distribution; Cl: clearance; PPB: plasma protein binding;(EQN means that value was calculated using VD=(Cl*t1/2)/0.693)Primary Target and PDB code of Protein-Drug complexTargets from DrugCentral Links
MIRABEGRON

MIRABEGRON


ATC G04BD12

GENITO
TREATMENT OF OVERACTIVE BLADDER (OAB)
AGONIST OF BETA-3 ADRENERGIC RECEPTOR (AR)

ORAL

F 29 PERCENT

VD 1670 LITER

PPB 71 PERCENT

Cl 57 LITER / HOUR

HT 50 HOUR

SOLUBILITY PRACTICALLY INSOLUBLE IN WATER 0.082 MILLIGRAM / MILLILITER

BETA-3 ADRENERGIC RECEPTOR

BETA-3 ADRENERGIC RECEPTOR AGONIST CHEMBL246 BETA-3 ADRENERGIC RECEPTOR P13945 BETA-3 ADRENERGIC RECEPTOR HOMO SAPIENS MEMBRANE RECEPTOR 7TM1 SMALLMOL MONOAMINE RECEPTOR ADRENERGIC RECEPTOREMA

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