PASIREOTIDE | PASIREOTIDE | ATC H01CB05
HORMONES CUSHINGS DISEASE SOMATOSTATIN ANALOGUE HUMAN SOMATOSTATIN RECEPTORS (HSST) AGONISTS LEADS TO DECREASED CORTISOL SECRETION HSST1 (IC50 = 9.3 NANOMOLAR) HSST2 (IC50 = 1.0 NANOMOLAR) HSST3 (IC50 = 1.5 NANOMOLAR) HSST4 (IC50 > 1000 NANOMOLAR) HSST5 (IC50 = 0.16 NANOMOLAR) | SUBCUTANEOUS INTRAMUSCULAR | VD 100 LITER PPB 88 PERCENT Cl 7.6 LITER / HOUR HT 12 HOUR | SOMATOSTATIN RECEPTORS (SST) | SOMATOSTATIN RECEPTOR 1 AGONIST CHEMBL1917 SOMATOSTATIN RECEPTOR 1 P30872 SOMATOSTATIN RECEPTOR TYPE 1 HOMO SAPIENS MEMBRANE RECEPTOR 7TM1 PEPTIDE SHORT PEPTIDE SOMATOSTATIN RECEPTOR | EMA ANSM (in French) Inxight Drugs Dailymed Drugs.com SIDER side effects Chemical Probes Portal ChEMBL BindingDB DrugBank |