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1 INNClassRoute (list)PK parameters= Cmax; Tmax; F: bioavailability; t1/2: half-life; VD: volume of distribution; Cl: clearance; PPB: plasma protein binding;(EQN means that value was calculated using VD=(Cl*t1/2)/0.693)Primary Target and PDB code of Protein-Drug complexTargets from DrugCentral Links
LOMITAPIDE

LOMITAPIDE


ATC C10AX12

CARDIOVASCULAR
INHIBITOR OF MICROSOMAL TRIGLYCERIDE TRANSFER PROTEIN (MTP) AND REDUCED LEVELS OF PLASMA LDL-C

ORAL

F 7 PERCENT

VD 1138 LITER

PPB 99.8 PERCENT

Cl 19.8 LITER / HOUR (EQN)

HT 39.7 HOUR

SOLUBILITY SLIGHTLY SOLUBLE IN AQUEOUS SOLUTIONS OF PH 2 TO 5

MICROSOMAL TRIGLYCERIDE TRANSFER PROTEIN

MICROSOMAL TRIGLYCERIDE TRANSFER PROTEIN INHIBITOR CHEMBL2364681 MICROSOMAL TRIGLYCERIDE TRANSFER PROTEIN P55157 MICROSOMAL TRIGLYCERIDE TRANSFER PROTEIN LARGE SUBUNIT HOMO SAPIENS CYTOSOLIC OTHEREMA

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