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1 INNClassRoute (list)PK parameters= Cmax; Tmax; F: bioavailability; t1/2: half-life; VD: volume of distribution; Cl: clearance; PPB: plasma protein binding;(EQN means that value was calculated using VD=(Cl*t1/2)/0.693)Primary Target and PDB code of Protein-Drug complexTargets from DrugCentral Links
M AZILSARTAN KAMEDOXOMIL (is an active metabolite)

AZILSARTAN KAMEDOXOMIL


ATC C09CA09
ATC C09DA09

CARDIOVASCULAR
ANTIHYPERTENSIVE
ANGIOTENSIN II RECEPTOR BLOCKER
SELECTIVE AT1 SUBTYPE ANGIOTENSIN II RECEPTOR ANTAGONIST

-

Tmax 2.25 HOUR

F 60 PERCENT

VD 16 LITER

PPB 99 PERCENT

Cl 0.138 LITER / HOUR

HT 11 HOUR

AT1 RECEPTOR

Type-1 angiotensin II receptor P30556 (AGTR1_HUMAN)EMA

ANSM (in French)

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