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1 INNClassRoute (list)PK parameters= Cmax; Tmax; F: bioavailability; t1/2: half-life; VD: volume of distribution; Cl: clearance; PPB: plasma protein binding;(EQN means that value was calculated using VD=(Cl*t1/2)/0.693)Primary Target and PDB code of Protein-Drug complexTargets from DrugCentral Links
INDACATEROL DISCONTINUED

INDACATEROL


ATC R03AC18
ATC R03AL04
ATC R03AK14
ATC R03AL12

RESPIRATORY
BRONCHODILATOR
SELECTIVE BETA2 ADRENERGIC AGONIST
CHRONIC OBSTRUCTIVE PULMONARY DISEASE (COPD)

INHALATION

F 44 PERCENT

VD 2459 LITER

PPB 95 PERCENT

Cl 21.05 LITER / HOUR

HT 85.7 HOUR

SOLUBILITY VERY SLIGHTLY SOLUBLE IN WATER

BETA-2-ADRENORECEPTOR

BETA-2 ADRENERGIC RECEPTOR AGONIST CHEMBL210 BETA-2 ADRENERGIC RECEPTOR P07550 BETA-2 ADRENERGIC RECEPTOR HOMO SAPIENS MEMBRANE RECEPTOR 7TM1 SMALLMOL MONOAMINE RECEPTOR ADRENERGIC RECEPTOREMA

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