RUFINAMIDE | RUFINAMIDE | ATC N03AF03
NERVOUS SYSTEM ANTIEPILEPTIC PROLONGATION OF THE INACTIVE STATE OF THE CHANNEL INHIBITOR | ORAL | Tmax 5 HOUR F 85 PERCENT (600 MILLIGRAM) VD 50 LITER (3200 MILLIGRAM / DAY) PPB 34 PERCENT Cl 4.3 LITER / HOUR (EQN) HT 8 HOUR SOLUBILITY PRACTICALLY INSOLUBLE IN WATER | SODIUM CHANNELS (EC50 = 3.8 MICROMOLAR) | SODIUM CHANNEL ALPHA SUBUNIT BLOCKER CHEMBL2331043 SODIUM CHANNEL ALPHA SUBUNIT P35498 SODIUM CHANNEL PROTEIN TYPE 1 SUBUNIT ALPHA HOMO SAPIENS ION CHANNEL VGC VG NA | EMA ANSM (in French) Inxight Drugs Dailymed Drugs.com SIDER side effects Chemical Probes Portal ChEMBL BindingDB DrugBank |