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1 INNClassRoute (list)PK parameters= Cmax; Tmax; F: bioavailability; t1/2: half-life; VD: volume of distribution; Cl: clearance; PPB: plasma protein binding;(EQN means that value was calculated using VD=(Cl*t1/2)/0.693)Primary Target and PDB code of Protein-Drug complexTargets from DrugCentral Links
SALMETEROL

SALMETEROL


ATC R03AC12
ATC R03AK06
ATC R03AK12

RESPIRATORY
SYMPATHOMIMETIC
BETA2-ADRENERGIC BRONCHODILATOR AGONIST

INHALATION

Cmax 0.36 NANOMOLAR (42 MICROGRAM TWICE DAILY)

PPB 96 PERCENT

HT 5.5 HOUR

SOLUBILITY SPARINGLY SOLUBLE IN WATER

BETA-2 ADRENERGIC RECEPTOR

BETA-2 ADRENERGIC RECEPTOR AGONIST CHEMBL210 BETA-2 ADRENERGIC RECEPTOR P07550 BETA-2 ADRENERGIC RECEPTOR HOMO SAPIENS MEMBRANE RECEPTOR 7TM1 SMALLMOL MONOAMINE RECEPTOR ADRENERGIC RECEPTOREMA

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