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1 INNClassRoute (list)PK parameters= Cmax; Tmax; F: bioavailability; t1/2: half-life; VD: volume of distribution; Cl: clearance; PPB: plasma protein binding;(EQN means that value was calculated using VD=(Cl*t1/2)/0.693)Primary Target and PDB code of Protein-Drug complexTargets from DrugCentral Links
SUFENTANIL

SUFENTANIL


ATC N01AH03

NERVOUS SYSTEM
ANALGESIC
ANESTHETICS
NARCOTICS
OPIATE AGONISTS

INJECTION SUBLINGUAL

Cmax 0.26 NANOMOLAR

VD 611 LITER (65 KILOGRAM)

PPB 93 PERCENT

Cl 58.5 LITER / HOUR (65 KILOGRAM)

HT 2.7 HOUR

MU-TYPE OPIOID RECEPTOR

MU OPIOID RECEPTOR AGONIST CHEMBL233 MU OPIOID RECEPTOR P35372 MU-TYPE OPIOID RECEPTOR HOMO SAPIENS MEMBRANE RECEPTOR 7TM1 PEPTIDE SHORT PEPTIDE OPIOID RECEPTOREMA

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