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1 INNClassRoute (list)PK parameters= Cmax; Tmax; F: bioavailability; t1/2: half-life; VD: volume of distribution; Cl: clearance; PPB: plasma protein binding;(EQN means that value was calculated using VD=(Cl*t1/2)/0.693)Primary Target and PDB code of Protein-Drug complexTargets from DrugCentral Links
PINDOLOL

PINDOLOL


ATC C07AA03
ATC C07CA03

CARDIOVASCULAR
ANTIHYPERTENSIVE AGENTS
NON SELECTIVE BETA ADRENERGIC RECEPTOR ANTAGONISTS
VASODILATOR AGENTS
SYMPATHOMIMETIC

ORAL

Cmax 427 NANOMOLAR

Tmax 1 HOUR

F 95 PERCENT

VD 130 LITER (65 KILOGRAM)

PPB 40 PERCENT

Cl 30 LITER / HOUR

HT 3.5 HOUR

SOLUBILITY SOLUBLE IN AQUAEOUS ACIDS

BETA ADRENERGIC RECEPTOR

BETA-2 ADRENERGIC RECEPTOR PARTIAL AGONIST CHEMBL210 BETA-2 ADRENERGIC RECEPTOR P07550 BETA-2 ADRENERGIC RECEPTOR HOMO SAPIENS MEMBRANE RECEPTOR 7TM1 SMALLMOL MONOAMINE RECEPTOR ADRENERGIC RECEPTOREMA

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