e-Drug3D

954

RETAPAMULIN

DISCONTINUED

INN
RETAPAMULIN

cas 224452-66-8

CLASS

DERMATOLOGICALS
ANTIBACTERIAL
A SEMISYNTHETIC PLEUROMUTILIN ANTIBIOTIC

ROUTE (list)

TOPICAL

ATC code

D06AX13

PK parameters

PPB 94 PERCENT

Target

TARGET 50S RIBOSOMAL PROTEIN L3

DrugCentral

Unknown

Download SDF file

Acetic acid, 2-[[(3-exo)-8-methyl-8-azabicyclo[3.2.1]oct-3-yl]thio]-, (3aS,4R,5S,6S,8R,9R,9aR,10R)-6-ethenyldecahydro-5-hydroxy-4,6,9,10-tetramethyl-1-oxo-3a,9-propano-3aH-cyclopentacycloocten-8-yl ester

Formula:
C30H47NO4S

Calculated chemical properties:

MW 517.76
NB_atoms 36
XLogP 5.25
PSA 64.118
NB_HD 1
NB_HA 5
fsp3 0.87
Lipinski(0=no;1=yes) 0

FDA
NDA 022055 (label) INN (RETAPAMULIN) ALTABAX (ALMIRALL) APPROVAL= AP YEAR= 2007 NEWMOLECULARENTITY DISCONTINUED