e-Drug3D

709

HALOFANTRINE

DISCONTINUED

INN
HALOFANTRINE

cas 69756-53-2

CLASS

ANTIPARASITIC
ANTIMALARIAL
SCHIZONTICIDAL ANTIMALARIAL AGENT

ROUTE (list)

ORAL

ATC code

P01BX01

PK parameters

t1/2 192 HOUR

Solubility

PRATICALLY INSOLUBLE IN WATER

Target

TARGET FERRIPROTOPORPHYRIN IX (FE(III)PPIX) (PMID18508124)

Unknown

Download SDF file

3-(dibutylamino)-1-[1,3-dichloro-6-(trifluoromethyl)phenanthren-9-yl]propan-1-ol

Formula:
C26H30Cl2F3NO

Calculated chemical properties:

MW 500.41
NB_atoms 33
XLogP 8.64
PSA 23.888
NB_HD 1
NB_HA 2
fsp3 0.46
Lipinski(0=no;1=yes) 0

FDA
NDA 020250 (label) INN (HALOFANTRINE HYDROCHLORIDE) HALFAN (GLAXOSMITHKLINE) APPROVAL= AP YEAR= 1992 DISCONTINUED