e-Drug3D

571

DEZOCINE

DISCONTINUED

INN
DEZOCINE

cas 53648-55-8

CLASS

NERVOUS SYSTEM
NARCOTIC ANTAGONIST
ANALGESIC OPIOD

ROUTE (list)

INJECTION

ATC code

N02AX03

PK parameters

Tmax 0.03 HOUR
VD 390 LITER (65 KILOGRAM)
Cl 97.5 LITER / HOUR (65 KILOGRAM)
PPB 91.6 PERCENT
t1/2 4 HOUR

Target

TARGET KAPPA-TYPE OPIOID RECEPTOR
MU-TYPE OPIOID RECEPTOR

Mu-type opioid receptor UNIPROT P35372 OPRM1

Kappa-type opioid receptor UNIPROT P41145 OPRK1

Download SDF file

5,11-Methanobenzocyclodecen-3-ol, 13-amino-5,6,7,8,9,10,11,12-octahydro-5-methyl-, (5R,11S,13S)-

Formula:
C16H23NO

Calculated chemical properties:

MW 245.35
NB_atoms 18
XLogP 3.11
PSA 41.714
NB_HD 3
NB_HA 2
fsp3 0.62
Lipinski(0=no;1=yes) 1

FDA
NDA 019082 (pdf not found) INN (DEZOCINE) DALGAN (ASTRAZENECA) APPROVAL= - YEAR= 0 DISCONTINUED