e-Drug3D

356

cas 548-73-2

CLASS

NERVOUS SYSTEM
ANTIPSYCHOTIC
ANESTHESIA
ANTIEMETICS
DOPAMINE ANTAGONISTS
A NEUROLEPTIC (TRANQUILIZER) AGENT

ROUTE (list)

INJECTION

PK parameters

VD 103 LITER
Cl 44 LITER / HOUR (PMID3179149)
t1/2 2.1 HOUR

TARGET D(2) DOPAMINE RECEPTOR

PDB
6X6G (CRYSTAL STRUCTURE OF ACETYLTRANSFERASE EIS FROM MYCOBACTERIUM TUBERCULOSIS IN COMPLEX WITH DROPERIDOL)

Ligand code = USS (link to the list of PDB complexes)

Download experimental 3D coordinates of USS with added hydrogens

MW 379.43
NB_atoms 28
XLogP 3.68
PSA 53.441
NB_HD 1
NB_HA 5
fsp3 0.27
Lipinski(0=no;1=yes) 1

FDA
NDA 016049 (pdf not found) INN (DROPERIDOL ; FENTANYL CITRATE) INNOVAR (EPIC PHARMA LLC) APPROVAL= - YEAR= 0 DISCONTINUED
NDA 071754 (pdf not found) INN (DROPERIDOL) DROPERIDOL (SOLOPAK) APPROVAL= - YEAR= 0 DISCONTINUED
NDA 071755 (pdf not found) INN (DROPERIDOL) DROPERIDOL (SOLOPAK) APPROVAL= - YEAR= 0 DISCONTINUED
NDA 071941 (pdf not found) INN (DROPERIDOL) DROPERIDOL (QUAD PHARMS) APPROVAL= - YEAR= 0 DISCONTINUED
NDA 071942 (pdf not found) INN (DROPERIDOL) DROPERIDOL (QUAD PHARMS) APPROVAL= - YEAR= 0 DISCONTINUED
NDA 072020 (pdf not found) INN (DROPERIDOL) DROPERIDOL (IGI LABS INC) APPROVAL= - YEAR= 0 DISCONTINUED
NDA 072026 (pdf not found) INN (DROPERIDOL ; FENTANYL CITRATE) FENTANYL CITRATE AND DROPERIDOL (ASTRAZENECA) APPROVAL= - YEAR= 0 DISCONTINUED
NDA 072027 (pdf not found) INN (DROPERIDOL ; FENTANYL CITRATE) FENTANYL CITRATE AND DROPERIDOL (ASTRAZENECA) APPROVAL= - YEAR= 0 DISCONTINUED
NDA 072028 (pdf not found) INN (DROPERIDOL ; FENTANYL CITRATE) FENTANYL CITRATE AND DROPERIDOL (ASTRAZENECA) APPROVAL= - YEAR= 0 DISCONTINUED
NDA 073520 (pdf not found) INN (DROPERIDOL) DROPERIDOL (WATSON LABS) APPROVAL= - YEAR= 0 DISCONTINUED
NDA 073521 (pdf not found) INN (DROPERIDOL) DROPERIDOL (WATSON LABS) APPROVAL= - YEAR= 0 DISCONTINUED
NDA 073523 (pdf not found) INN (DROPERIDOL) DROPERIDOL (WATSON LABS) APPROVAL= - YEAR= 0 DISCONTINUED
NDA 016796 (pdf not found) INN (DROPERIDOL) INAPSINE (RISING) APPROVAL= AP YEAR= 1970 DISCONTINUED
NDA 070992 (pdf not found) INN (DROPERIDOL) DROPERIDOL (ABRAXIS PHARM) APPROVAL= AP YEAR= 1986 DISCONTINUED
NDA 070993 (pdf not found) INN (DROPERIDOL) DROPERIDOL (ABRAXIS PHARM) APPROVAL= AP YEAR= 1986 DISCONTINUED
NDA 071645 (pdf not found) INN (DROPERIDOL) DROPERIDOL (HOSPIRA) APPROVAL= AP YEAR= 1988 DISCONTINUED
NDA 071750 (pdf not found) INN (DROPERIDOL) DROPERIDOL (SMITH AND NEPHEW) APPROVAL= AP YEAR= 1988 DISCONTINUED
NDA 071981 (pdf not found) INN (DROPERIDOL) DROPERIDOL (HOSPIRA) APPROVAL= AP YEAR= 1988 DISCONTINUED
NDA 071982 (pdf not found) INN (DROPERIDOL ; FENTANYL CITRATE) FENTANYL CITRATE AND DROPERIDOL (HOSPIRA) APPROVAL= AP YEAR= 1988 DISCONTINUED
NDA 072018 (pdf not found) INN (DROPERIDOL) DROPERIDOL (ASTRAZENECA) APPROVAL= AP YEAR= 1988 DISCONTINUED
NDA 072019 (pdf not found) INN (DROPERIDOL) DROPERIDOL (IGI LABS INC) APPROVAL= AP YEAR= 1988 DISCONTINUED
NDA 072021 (pdf not found) INN (DROPERIDOL) DROPERIDOL (IGI LABS INC) APPROVAL= AP YEAR= 1988 DISCONTINUED
NDA 072123 (pdf not found) INN (DROPERIDOL) DROPERIDOL (AM REGENT) APPROVAL= AP YEAR= 1988
NDA 072335 (pdf not found) INN (DROPERIDOL) DROPERIDOL (LUITPOLD) APPROVAL= AP YEAR= 1988 DISCONTINUED
NDA 072272 (pdf not found) INN (DROPERIDOL) DROPERIDOL (HOSPIRA) APPROVAL= AP YEAR= 1995 DISCONTINUED
NDA 208197 (pdf not found) INN (DROPERIDOL) DROPERIDOL (HIKMA) APPROVAL= AP YEAR= 2017